Nek2 inhibitor 72

CAS No. ——

Nek2 inhibitor 72( —— )

Catalog No. M17076 CAS No. ——

A potent, ATP-competitive and relative selective Nek2 inhibitor with IC50 of 0.27 uM.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    Nek2 inhibitor 72
  • Note
    Research use only, not for human use.
  • Brief Description
    A potent, ATP-competitive and relative selective Nek2 inhibitor with IC50 of 0.27 uM.
  • Description
    A potent, ATP-competitive and relative selective Nek2 inhibitor with IC50 of 0.27 uM; displays >10-fold selectivity over CDK2.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    ——
  • Pathway
    Cell Cycle/DNA Damage
  • Target
    Hec1/Nek2
  • Recptor
    Hec1/Nek2
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    ——
  • Formula Weight
    334.427
  • Molecular Formula
    C19H22N6
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    ——
  • Chemical Name
    (E)-6-(2-(azepan-1-yl)vinyl)-N-phenyl-9H-purin-2-amine

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Coxon CR, et al. Oncotarget. 2017 Mar 21;8(12):19089-19124.
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